Fast assembly of 1 H -imidazo[1,2- a ]imidazol-5-amines via groebke-blackburn-bienaymé reaction with 2-aminoimidazoles

Olga P. Pereshivko, Vsevolod A. Peshkov, Denis S. Ermolat'Ev, Erik V. Van Der Eycken

Research output: Contribution to journal › Article

15 Citations (Scopus)

Abstract

A novel microwave-assisted protocol allowing the successful application of 2-aminoimidazoles in the Groebke-Blackburn-Bienaymé reaction for the facile construction of the 1H-imidazo[1,2-a]imidazol-5-amine core was developed.

Original languageEnglish
Article numberST-2012-B0834-L
Pages (from-to)351-354
Number of pages4
JournalSynlett
Volume24
Issue number3
DOIs
Publication statusPublished - Jan 17 2013
Externally publishedYes

Fingerprint

Amines
Microwaves
2-aminoimidazole

Keywords

  • annulation
  • fused-ring systems
  • heterocycles
  • multicomponent reactions

ASJC Scopus subject areas

  • Organic Chemistry

Cite this

Fast assembly of 1 H -imidazo[1,2- a ]imidazol-5-amines via groebke-blackburn-bienaymé reaction with 2-aminoimidazoles. / Pereshivko, Olga P.; Peshkov, Vsevolod A.; Ermolat'Ev, Denis S.; Van Der Eycken, Erik V.

In: Synlett, Vol. 24, No. 3, ST-2012-B0834-L, 17.01.2013, p. 351-354.

Research output: Contribution to journal › Article

Pereshivko, OP, Peshkov, VA, Ermolat'Ev, DS & Van Der Eycken, EV 2013, 'Fast assembly of 1 H -imidazo[1,2- a ]imidazol-5-amines via groebke-blackburn-bienaymé reaction with 2-aminoimidazoles', Synlett, vol. 24, no. 3, ST-2012-B0834-L, pp. 351-354. https://doi.org/10.1055/s-0032-1317986
Pereshivko OP, Peshkov VA, Ermolat'Ev DS, Van Der Eycken EV. Fast assembly of 1 H -imidazo[1,2- a ]imidazol-5-amines via groebke-blackburn-bienaymé reaction with 2-aminoimidazoles. Synlett. 2013 Jan 17;24(3):351-354. ST-2012-B0834-L. https://doi.org/10.1055/s-0032-1317986
Pereshivko, Olga P. ; Peshkov, Vsevolod A. ; Ermolat'Ev, Denis S. ; Van Der Eycken, Erik V. / Fast assembly of 1 H -imidazo[1,2- a ]imidazol-5-amines via groebke-blackburn-bienaymé reaction with 2-aminoimidazoles. In: Synlett. 2013 ; Vol. 24, No. 3. pp. 351-354.
@article{d59acf4dd6c14d9fba4285f67a0f3a24,
title = "Fast assembly of 1 H -imidazo[1,2- a ]imidazol-5-amines via groebke-blackburn-bienaym{\'e} reaction with 2-aminoimidazoles",
abstract = "A novel microwave-assisted protocol allowing the successful application of 2-aminoimidazoles in the Groebke-Blackburn-Bienaym{\'e} reaction for the facile construction of the 1H-imidazo[1,2-a]imidazol-5-amine core was developed.",
keywords = "annulation, fused-ring systems, heterocycles, multicomponent reactions",
author = "Pereshivko, {Olga P.} and Peshkov, {Vsevolod A.} and Ermolat'Ev, {Denis S.} and {Van Der Eycken}, {Erik V.}",
year = "2013",
month = "1",
day = "17",
doi = "10.1055/s-0032-1317986",
language = "English",
volume = "24",
pages = "351--354",
journal = "Synlett",
issn = "0936-5214",
publisher = "Georg Thieme Verlag",
number = "3",

}

TY - JOUR

T1 - Fast assembly of 1 H -imidazo[1,2- a ]imidazol-5-amines via groebke-blackburn-bienaymé reaction with 2-aminoimidazoles

AU - Pereshivko, Olga P.

AU - Peshkov, Vsevolod A.

AU - Ermolat'Ev, Denis S.

AU - Van Der Eycken, Erik V.

PY - 2013/1/17

Y1 - 2013/1/17

N2 - A novel microwave-assisted protocol allowing the successful application of 2-aminoimidazoles in the Groebke-Blackburn-Bienaymé reaction for the facile construction of the 1H-imidazo[1,2-a]imidazol-5-amine core was developed.

AB - A novel microwave-assisted protocol allowing the successful application of 2-aminoimidazoles in the Groebke-Blackburn-Bienaymé reaction for the facile construction of the 1H-imidazo[1,2-a]imidazol-5-amine core was developed.

KW - annulation

KW - fused-ring systems

KW - heterocycles

KW - multicomponent reactions

UR - http://www.scopus.com/inward/record.url?scp=84872200100&partnerID=8YFLogxK

UR - http://www.scopus.com/inward/citedby.url?scp=84872200100&partnerID=8YFLogxK

U2 - 10.1055/s-0032-1317986

DO - 10.1055/s-0032-1317986

M3 - Article

AN - SCOPUS:84872200100

VL - 24

SP - 351

EP - 354

JO - Synlett

JF - Synlett

SN - 0936-5214

IS - 3

M1 - ST-2012-B0834-L

ER -

Access to Document