@article{250edccea75443c1b6fb8b86859d9270,
title = "Gold-catalyzed post-Ugi alkyne hydroarylation for the synthesis of 2-quinolones",
abstract = "A series of propargylamides containing an electron-rich benzene ring was prepared through the Ugi reaction of 3,5-dimethoxy-aniline with various propiolic acids, aldehydes and isocyanides. Subjecting these adducts to a gold-catalyzed intramolecular alkyne hydroarylation process allowed to efficiently construct the 2-quinolone core bearing a branched substituent on the nitrogen atom.",
keywords = "2-quinolones, Gold catalysis, Hydroarylation, Ugi reaction",
author = "Xiaochen Du and Jianjun Huang and Nechaev, {Anton A.} and Ruwei Yao and Jing Gong and {Van Der Eycken}, {Erik V.} and Pereshivko, {Olga P.} and Peshkov, {Vsevolod A.}",
note = "Funding Information: This work was supported by the start-up fund from Soochow University (grant Q410900714), National Natural Science Foundation of China (grant 21650110445), Natural Science Foundation of Jiangsu Province of China (grants BK20160310and BK20150317), the Priority Academic Program Development of Jiangsu Higher Education Institutions (PAPD) and the project of scientific and technologic infrastructure of Suzhou (grant SZS201708). A. A. N. is grateful to the European Community Mobility Programme “Erasmus Mundus Action 2, Strand 1” for providing a doctoral scholarship. E. V. V. d. E. acknowledges the support of RUDN University Program 5-100.",
year = "2018",
month = oct,
day = "4",
doi = "10.3762/bjoc.14.234",
language = "English",
volume = "14",
pages = "2572--2579",
journal = "Beilstein Journal of Organic Chemistry",
issn = "1860-5397",
publisher = "Beilstein-Institut Zur Forderung der Chemischen Wissenschaften",
}